APINACA
 | |
| Material name by the IUPAC glossology | |
|---|---|
| 1-pentyl group-N-bird chloro[3,3,1,13,7]dec-1-yl-1H- indazole-3-carboxamide | |
| Clinical data | |
| Legal regulation |
|
| Identification | |
| CAS number (MeSH) | 1,345,973-53-6 |
| ChemSpider | 28189076 |
| Chemical data | |
| Chemical formula | C23H31N3O |
| Molecular weight | 365.510 |
| |
| |
AKB48) is an agonist of cannabinoids 1 receptor (CB1R) [1] APINACA (N-(1-adamantyl)-1-pentyl-1H-indazole-3-carboxamide, a common name (Ki=304.5nM, EC50=585nM).
I was confirmed as an ingredient of the dangerous herb (synthetic cannabinoids) like APICA () at a research institute of Japan in March, 2012 [2]. In Japan, was added to a designated drug based on the Drugs, Cosmetics and Medical Instruments Act on July 1, 2012, and was said that was illegal [3]; [4] [5]. In addition, in the New Zealand, I was appointed in a designated drug (Temporary class drug) at one time on July 13, 2012 and was forbidden [6].
It is kind of synthetic cannabinoids and is the compound which a pentyl group connected to the first place of indazole. It was within the range applied to a certain patent for, but this compound in itself has not been listed in an article and a patent [7].
Table of contents
Detection
May be sold by a name AKB48 with the drug [8]; [9]. The law standard of the medicine machine method is effective in this drug. I am listed by the drug which there is possibility of the abuse in in a website of フォレンデックス (Forendex) [10].
Allied item
Footnote
- ^ Uchiyama, N.; Kawamura, M.; Kikura-Hanajiri, R.; Goda, Y. (2012). "URB-754: A new class of designer drug and 12 synthetic cannabinoids detected in illegal products." Forensic Science International 227 (1–3): 21–32. doi: 10.1016/j.forsciint.2012.08.047. PMID 23063179.
- ^ Uchiyama, N.; Kawamura, M.; Kikura-Hanajiri, R.; Goda, Y. (2012). "Identification of two new-type synthetic cannabinoids, N-(1-adamantyl)-1-pentyl-1H-indole-3-carboxamide (APICA) and N-(1-adamantyl)-1-pentyl-1H-indazole-3-carboxamide (APINACA), and detection of five synthetic cannabinoids, AM-1220, AM-2233, AM-1241, CB-13 (CRA-13), and AM-1248, as designer drugs in illegal products." Forensic Toxicology 30 (2): 114. doi: 10.1007/s11419-012-0136-7.
- ^ "About revision of the departmental order to establish uses such as the medical care to prescribe to 4 of designated drug to prescribe in the Drugs, Cosmetics and Medical Instruments Act Article 2 Clause 14 and law Article 76 (notice of enforcement) (PDF)". Ministry of Health, Labour and Welfare medicine food chief of the bureau (June 1, 2012). September 23, 2012 reading.
- For designated (substance regulated) 1,960 years of "the designated drug" by the rule of ^ the Drugs, Cosmetics and Medical Instruments Act, it is law 145th
- List of ^ designation drugs - Ministry of Health, Labour and Welfare
- ^ Temporary Class Drug Notice, 05 July 2012. NZ Department of Internal Affairs. - The New Zealand government
- ^ patent WO 2003/035005
- ^ Federal Register Volume 78, Number 71 (Friday, April 12, 2013)
- ^ AKB48 (APINACA) and 5F-AKB48 (5F-APINACA) DEA/OD/ODE (May, 2013)
- ^ SAFS | Forendex
Outside link
This article is taken from the Japanese Wikipedia APINACA
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